1. Signaling Pathways
  2. Antibody-drug Conjugate/ADC Related
  3. ADC Cytotoxin
  4. ADC Cytotoxin Inhibitors

ADC Cytotoxin Inhibitors

Auristatin

Calicheamicins

Camptothecins

Daunorubicins/Doxorubicins

Duocarmycins

Maytansinoids

Pyrrolobenzodiazepines

Traditional Cytotoxic Agents

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ADC Cytotoxin
Product Name Auristatin Calicheamicins Camptothecins Daunorubicins/Doxorubicins Duocarmycins Maytansinoids Pyrrolobenzodiazepines Traditional Cytotoxic Agents Purity
Doxorubicin hydrochloride      
Daunorubicins/Doxorubicins
        99.90%
Paclitaxel              
Traditional Cytotoxic Agents
99.97%
Monomethyl auristatin E
Auristatin
              99.97%
Exatecan mesylate    
Camptothecins
          99.92%
(αR)-Cyclopropaneacetamide-Exatecan    
Camptothecins
          99.75%
Dxd    
Camptothecins
          ≥99.0%
SN-38    
Camptothecins
          99.89%
Methotrexate              
Traditional Cytotoxic Agents
99.75%
Camptothecin    
Camptothecins
          99.82%
Mertansine          
Maytansinoids
    99.80%
Daunorubicin hydrochloride      
Daunorubicins/Doxorubicins
        99.62%
Exatecan    
Camptothecins
          99.93%
MMAF
Auristatin
              99.91%
Exatecan Intermediate 1    
Camptothecins
          99.99%
α-Amanitin              
Traditional Cytotoxic Agents
99.92%
MMAE-d8
Auristatin
              99.29%
Exatecan-d5 mesylate    
Camptothecins
          99.82%
Calicheamicin  
Calicheamicins
            98.28%
SG3199            
Pyrrolobenzodiazepines
  98.94%
Aldoxorubicin      
Daunorubicins/Doxorubicins
       
PNU-159682      
Daunorubicins/Doxorubicins
        98.25%
(4-NH2)-Exatecan    
Camptothecins
          ≥99.0%
Exatecan Intermediate 2    
Camptothecins
          99.95%
Taltobulin              
Traditional Cytotoxic Agents
99.90%
Auristatin E
Auristatin
              99.75%
SJG-136            
Pyrrolobenzodiazepines
  99.43%
MMAF hydrochloride
Auristatin
              99.52%
Duocarmycin TM        
Duocarmycins
      98.04%
Exatecan Intermediate 6    
Camptothecins
          98.92%
PF-06380101
Auristatin
              99.47%
Duocarmycin DM free base      
Daunorubicins/Doxorubicins
        98.11%
Ansamitocin P-3          
Maytansinoids
    ≥98.0%
Dolastatin 10
Auristatin
              98.11%
Daun02      
Daunorubicins/Doxorubicins
        98.72%
β-Amanitin              
Traditional Cytotoxic Agents
SG2057            
Pyrrolobenzodiazepines
  98.67%
MMAF-d8 hydrochloride
Auristatin
              99.70%
MMAD
Auristatin
              99.94%
(R)-Exatecan Intermediate 1    
Camptothecins
         
MMAF-OMe
Auristatin
              99.62%
Fmoc-MMAE
Auristatin
              99.20%
DM3          
Maytansinoids
   
Tubulysin A              
Traditional Cytotoxic Agents
99.08%
Duocarmycin SA        
Duocarmycins
      ≥98.0%
MMAF sodium
Auristatin
              99.62%
DC0-NH2        
Duocarmycins
     
DM1-SMe          
Maytansinoids
    98.02%
DM4-SMe          
Maytansinoids
    ≥98.0%
Tomaymycin DM            
Pyrrolobenzodiazepines
  98.01%
(1R,9R)-Exatecan mesylate    
Camptothecins
          99.94%
10-Deacetyl-7-xylosyl paclitaxel              
Traditional Cytotoxic Agents
99.65%
Ac-Exatecan    
Camptothecins
          98.70%
Exatecan-amide-cyclopropanol    
Camptothecins
          98.15%
Hemiasterlin            
Pyrrolobenzodiazepines
  99.77%
Cyclopropaneacetamide-Exatecan    
Camptothecins
         
(1S,9R)-Exatecan mesylate    
Camptothecins
         
PNU-159682 carboxylic acid      
Daunorubicins/Doxorubicins
       
Taltobulin hydrochloride              
Traditional Cytotoxic Agents
98.34%
(rac)-Exatecan Intermediate 1    
Camptothecins
          99.84%
PF-06380101-d8
Auristatin
              99.37%
Duocarmycin Analog        
Duocarmycins
     
DC1SMe        
Duocarmycins
      ≥98.0%
Exatecan-methylacetamide-OH    
Camptothecins
         
γ-Amanitin              
Traditional Cytotoxic Agents
Doxorubicin      
Daunorubicins/Doxorubicins
       
S-methyl DM1          
Maytansinoids
    99.58%
N-Me-L-Ala-maytansinol          
Maytansinoids
    99.89%
Taltobulin trifluoroacetate              
Traditional Cytotoxic Agents
99.08%
Exatecan Intermediate 5    
Camptothecins
          99.21%
Daunorubicin      
Daunorubicins/Doxorubicins
       
Exatecan Intermediate 7    
Camptothecins
          99.24%
Exatecan mesylate dihydrate    
Camptothecins
         
Duocarmycin A        
Duocarmycins
     
Exatecan mesylate (GMP)    
Camptothecins
         
C-11              
Traditional Cytotoxic Agents
DC1        
Duocarmycins
     
(+)-CBI-CDPI1        
Duocarmycins
     
DM3-SMe          
Maytansinoids
   
Seco-Duocarmycin SA        
Duocarmycins
     
DMEA-PNU-159682      
Daunorubicins/Doxorubicins
       
DC41SMe        
Duocarmycins
     
(+)-CBI-CDPI2        
Duocarmycins
     
Duocarmycin MB        
Duocarmycins
     
DC41        
Duocarmycins
     
DC4SMe        
Duocarmycins
     
Duocarmycin DM      
Daunorubicins/Doxorubicins
       
Seco-Duocarmycin TM        
Duocarmycins
     
Methotrexate monohydrate              
Traditional Cytotoxic Agents
Aniline-MPB-amino-C3-PBD            
Pyrrolobenzodiazepines
 
Rebeccamycin              
Traditional Cytotoxic Agents
DC10SMe        
Duocarmycins
     
Daunorubicin citrate      
Daunorubicins/Doxorubicins
       
Dolastatin 15
Auristatin
             
Isofistularin-3              
Traditional Cytotoxic Agents
ε-Amanitin              
Traditional Cytotoxic Agents
Gly-Cyclopropane-Exatecan    
Camptothecins
         
Mensacarcin              
Traditional Cytotoxic Agents
Tubulysin IM-2              
Traditional Cytotoxic Agents
Duocarmycin GA        
Duocarmycins
     
Py-MPB-amino-C3-PBD            
Pyrrolobenzodiazepines
 
Top1 inhibitor 1    
Camptothecins
         
Exatecan-amide-bicyclo[1.1.1]pentan-1-ylmethanol    
Camptothecins
         
Tubulysin IM-3              
Traditional Cytotoxic Agents
Exatecan-amide-bicyclo[1.1.1]pentan-1-ol    
Camptothecins
         
MMAD-d8
Auristatin
              98.95%
17-AEP-GA              
Traditional Cytotoxic Agents
Polyketomycin              
Traditional Cytotoxic Agents
Azonafide-PEABA              
Traditional Cytotoxic Agents
(1-OH)-Exatecan    
Camptothecins
         
Decyclohexanamine-Exatecan    
Camptothecins
         
17-GMB-APA-GA              
Traditional Cytotoxic Agents
Exatecan analogue 1    
Camptothecins
         
NH2-methylpropanamide-Exatecan TFA    
Camptothecins
          99.80%
Tubulysin IM-1              
Traditional Cytotoxic Agents
Corixetan              
Traditional Cytotoxic Agents
Sandramycin              
Traditional Cytotoxic Agents
Exatecan intermediate 11    
Camptothecins
         
Exatecan intermediate 10    
Camptothecins
         
Exatecan Intermediate 4 dihydrochloride    
Camptothecins
          99.92%
Exatecan intermediate 8    
Camptothecins
         
Exatecan analog 36    
Camptothecins
          98.71%
Exatecan Intermediate 2 hydrochloride    
Camptothecins
          99.33%
Exatecan Intermediate 3    
Camptothecins
         
Exatecan intermediate 9    
Camptothecins
         
Exatecan-amide-CH2-O-CH2-CH2-OH    
Camptothecins
         
Exatecan Intermediate 4    
Camptothecins